baseline estimated glomerular filtration rate (eGFR)
Overview
Baseline estimated glomerular filtration rate (eGFR) is the kidney function measured before treatment begins or at entry to a study, derived from serum creatinine or another filtration marker together with patient characteristics. It is used across nephrology, cardiology, oncology and pharmacology to characterize renal status, stratify risk, and decide eligibility and dose. What makes the baseline value distinct from any later one is its role as a reference: subsequent measurements are interpreted as change from it, and the slope of that change — not any single reading — is what defines progression and what nephroprotection trials are powered to detect.
It matters in drug development because the kidney clears a large share of drugs and their metabolites. A patient's baseline eGFR predicts exposure to renally eliminated agents, so it enters population pharmacokinetic models as a covariate alongside body weight, body mass index, sex, race, age, disease status and formulation, and it sets the thresholds below which a dose is reduced or the drug withheld. It has served this role in the pharmacokinetic characterization of agents such as the myeloperoxidase inhibitor mitiperstat, studied in healthy volunteers and in patients with heart failure with preserved or mildly reduced ejection fraction (HFpEF/HFmrEF).
Its use as a risk stratifier follows from the close coupling of kidney and cardiovascular disease: reduced baseline eGFR predicts mortality and cardiovascular events independently of the kidney outcomes it more obviously anticipates, which is why it appears in trial eligibility criteria across therapeutic areas rather than only in nephrology. Two cautions attach to the baseline specifically. A single pre-treatment value can misrepresent stable function if taken during acute illness or volume depletion, and an early post-treatment fall in eGFR is not necessarily injury — agents that lower intraglomerular pressure produce a dip from baseline that precedes long-term preservation of function.
Recent Publications Summary
Recent publications involving baseline glomerular filtration rate (eGFR) primarily used it as a clinical baseline characteristic in studies of cancer treatment outcomes, especially in EGFR-mutant non-small cell lung cancer (NSCLC) and other oncology settings. In a real-world single-center analysis of patients with EGFR-mutant advanced NSCLC treated with EGFR tyrosine kinase inhibitors (TKIs), baseline clinical data were used to evaluate survival outcomes by TKI generation, although the abstract does not specify eGFR-stratified results 41454492Dec. Similarly, a study examining early loss of skeletal muscle, osimertinib trough concentrations, and treatment outcomes in advanced EGFR+ NSCLC incorporated baseline patient characteristics as part of its exposure–outcome analysis, but the abstract does not report eGFR-specific findings 41997038Apr.
Baseline eGFR also appears in the context of sequential and resistance-directed EGFR-targeted therapy. A case report of EGFR exon 19 deletion lung adenocarcinoma with later airway metastases described repeated molecular profiling and sequential EGFR TKI use, including osimertinib and gefitinib, to manage acquired resistance; baseline renal function assessment would be clinically relevant in such treatment planning, but no eGFR-related outcome was reported in the abstract 41125377Oct. In pancreatic ductal adenocarcinoma, studies of vertical pathway inhibition combined KRAS, EGFR, and STAT3 targeting to achieve durable tumor regression, and another report highlighted EGFR-mediated adaptive resistance to KRASG12D blockade; however, these abstracts do not provide baseline eGFR-specific data or analyses 42224594Jun41801133Mar.
Other recent publications focused on EGFR-directed therapeutics and mechanistic oncology studies rather than renal-function stratification. These included EGFR-targeting or EGFR/HER2 dual-inhibitory compounds, EGFR-specific aptamer-modified nanoparticles for photothermal therapy, and mechanistic work on EGFR-linked signaling in glioma and NSCLC 42237319Jun41875675Mar42206690May42348047Jun41966746Apr. Across these reports, baseline eGFR was not presented as a study endpoint, and no publication in the provided set reported eGFR-specific efficacy, safety, or pharmacokinetic conclusions.
What Changes, What Holds
1. Baseline eGFR remains a prognostic covariate rather than a new treatment determinant
REINFORCES Recent oncology analyses continue to treat baseline eGFR as part of routine clinical characterization, with no reported eGFR-stratified efficacy or safety signal to revise its role. That leaves the settled view intact: baseline kidney function is still mainly a background factor that may help interpret treatment outcomes, not a newly established driver of response in EGFR-mutant NSCLC 41454492Dec41997038Apr.
2. Renal assessment stays clinically relevant in sequential EGFR-targeted therapy, but no new eGFR-specific effect is shown
REINFORCES The case-based and mechanistic reports keep baseline renal function in the realm of practical treatment planning for EGFR-directed regimens, yet they do not add evidence that baseline eGFR itself changes resistance biology or outcome. What remains unchanged is the baseline account: eGFR is a supportive clinical metric, while the new work offers no direct renal-function result to alter that understanding 41125377Oct42224594Jun.
3. EGFR-directed oncology studies still do not establish baseline eGFR as an outcome variable
REINFORCES These mechanistic and therapeutic reports broaden the EGFR literature, but they leave the kidney-function question untouched. Because the Overview already frames baseline eGFR as a clinical covariate and not a target, the absence of eGFR-specific efficacy, safety, or pharmacokinetic findings simply reinforces that it remains a contextual measure rather than a central endpoint in these studies 42237319Jun41875675Mar.
baseline estimated glomerular filtration rate (egfr)
Background Contexts
In the literature, the biological baseline, pathological conditions, or disease models commonly surrounding baseline estimated glomerular filtration rate (egfr) are described as follows:
- lung cancer brain metastases (Disease) — 6 papers: PMIDs 42284116, 42237319, 42202477, 41997038, etc.
- Cancers (Clinical Metric) — 2 papers: PMIDs 42206690, 41176577
- glioma (Disease) — 2 papers: PMIDs 42348047, 41966746
- pancreatic ductal adenocarcinoma (Disease) — 2 papers: PMIDs 42224594, 41801133
- afatinib (Therapy) — 1 paper: PMIDs 41875675
- disease progression and resistance mechanisms (Other) — 1 paper: PMIDs 42202477
- human papilloma virus (Organism) — 1 paper: PMIDs 41980433
- Ocimum (Organism) — 1 paper: PMIDs 42236954
- Oral Melanoma (Disease) — 1 paper: PMIDs 42342053
- pancreatic/colorectal cancer (Disease) — 1 paper: PMIDs 41801133
- Psoralea corylifolia L. (Organism) — 1 paper: PMIDs 42334659
- recurrent cervical cancer (Disease) — 1 paper: PMIDs 41980433
Methodologies & Technologies Used
Researchers utilize the following experimental methods, imaging platforms, computational models, or biological reagents to study baseline estimated glomerular filtration rate (egfr):
- molecular docking studies (Technology) — 3 papers: PMIDs 42348047, 42236954, 41176577
- Network Pharmacology (Technology) — 3 papers: PMIDs 42348047, 42236954, 41966746
- CCK-8 assay (Technology) — 2 papers: PMIDs 41966746, 41176577
- MDA-MB-231 (Cell Line) — 2 papers: PMIDs 42334659, 41875675
- transcriptomic and metabolomic analyses (Technology) — 2 papers: PMIDs 42236954, 41966746
- (chemo)radiotherapy (Biological Process) — 1 paper: PMIDs 42342053
- 128 mitiperstat-treated participants (Organism) — 1 paper: PMIDs 42101107
- 2856 plasma samples (Clinical Metric) — 1 paper: PMIDs 42101107
- A549 lung cancer cells (Cell Line) — 1 paper: PMIDs 41875675
- A549 xenograft models (Cell Line) — 1 paper: PMIDs 41176577
- afatinib (Therapy) — 1 paper: PMIDs 42224594
- Aicardi-Goutières syndrome (Cell Line) — 1 paper: PMIDs 41176577
Molecular Interventions & Targets
The primary molecular pathways, regulatory genes, enzymes, or therapeutic agents actively targeted and manipulated in relation to baseline estimated glomerular filtration rate (egfr) include:
- KRAS (Gene) — 2 papers: PMIDs 42224594, 41801133
- osimertinib (Therapy) — 2 papers: PMIDs 42202477, 41997038
- acylhydrazone derivatives (Chemical) — 1 paper: PMIDs 41176577
- ADAM17 (Protein) — 1 paper: PMIDs 42342053
- Agrimonolide (Chemical) — 1 paper: PMIDs 42236954
- B-cell lymphoma 2 (Protein) — 1 paper: PMIDs 42342053
- bakuchiol (Chemical) — 1 paper: PMIDs 42334659
- BRAF gene (Gene) — 1 paper: PMIDs 42202477
- CCND1 (Gene) — 1 paper: PMIDs 42236954
- CD44/JAK2/STAT3 signaling pathway (Pathway) — 1 paper: PMIDs 42224594
- Chronic lung diseases (Disease) — 1 paper: PMIDs 42101107
- compound 10e (Chemical) — 1 paper: PMIDs 41875675
Observed Outcomes & Phenotypes
The phenotypic changes, physiological endpoints, or clinical metrics observed and measured in connection with baseline estimated glomerular filtration rate (egfr) include:
- MDA content (Clinical Metric) — 2 papers: PMIDs 42348047, 41966746
- reactive oxygen species (Chemical) — 2 papers: PMIDs 41966746, 41875675
- tumor cell apoptosis (Biological Process) — 2 papers: PMIDs 41966746, 41875675
- 111 DEGs (Gene) — 1 paper: PMIDs 42342053
- 263 human targets (Protein) — 1 paper: PMIDs 42236954
- 35 bioactive coumarins (Chemical) — 1 paper: PMIDs 42236954
- 59 coumarins (Chemical) — 1 paper: PMIDs 42236954
- ACSL4 (Protein) — 1 paper: PMIDs 42348047
- anti-proliferative, pro-apoptotic, and anti-metastatic role of bakuchiol (Biological Process) — 1 paper: PMIDs 42334659
- antitumor activity (Clinical Metric) — 1 paper: PMIDs 42237319
- apoptotic pathways (Biological Process) — 1 paper: PMIDs 41563668
- apparent central volume of distribution (Clinical Metric) — 1 paper: PMIDs 42101107
General Takeaways & Clinical Potentials
The high-level concepts, clinical translations, and overarching conclusions proposed in the research surrounding baseline estimated glomerular filtration rate (egfr) are summarized below:
- acquired resistance (Biological Process) — 1 paper: PMIDs 41125377
- advanced HPV16-associated cervical cancer (Disease) — 1 paper: PMIDs 41980433
- antineoplastic (Therapy) — 1 paper: PMIDs 41176577
- bakuchiol as a promising HSP90-targeting natural compound (Other) — 1 paper: PMIDs 42334659
- cancer and inflammatory diseases (Disease) — 1 paper: PMIDs 42236954
- Cancers (Clinical Metric) — 1 paper: PMIDs 42206690
- ClinicalTrials.gov: NCT02712372 (Other) — 1 paper: PMIDs 42101107
- combination drug (Therapy) — 1 paper: PMIDs 42224594
- coumarin-based functional foods (Other) — 1 paper: PMIDs 42236954
- covalent dual inhibitor of EGFR and HER-2 (Therapy) — 1 paper: PMIDs 41875675
- covalent inhibitors (Chemical) — 1 paper: PMIDs 42284116
- different mitiperstat development programs (Other) — 1 paper: PMIDs 42101107